Clin Pharmacol Ther. by RxPG google_page_url = document.location; , sitemap YouTube The medications known to be CYP3A4 inhibitors are summarized in the below table based on their class of medications and classifications.1,2,5,6 . Drugs metabolized by CYP3A4 are called CYP3A4 substrates. WŠd] €ã\àÙÉ"™Ñd0ìC[nٍ•%m«mLò闇d±‹Eò¨v$v¤s#‹¿ÃKfW_ý\}ýõW?½~ó]Õ|óMõíw¯«o¯ž?ûêQ Q7muuóü™¨ý¨Ô4ÖRUC3Õ]_]}Ôr?þ}¨Þ?>ÖTïé? Katzenmaier S, Markert C, Riedel KD, Burhenne J, Haefeli WE, Mikus G. Determining the time course of CYP3A4 inhibition by potent reversible and irreversible CYP3A4 inhibitors using a limited sampling strategy. google_ad_channel ="1397725367"; P450 inhibitors are drugs that decrease the activity of the enzyme causing drugs that are also metabolized by the P450 system to be metabolized at a decreased rate. µš³ìë©É°6Âëò … This is a really tough topic because there are literally thousands of drug interactions and we honestly can’t remember all of them. 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